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-Structure paper
Title | Potent Allosteric Dengue Virus NS5 Polymerase Inhibitors: Mechanism of Action and Resistance Profiling |
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Journal, issue, pages | Plos Pathog., Vol. 12, Page e1005737-e1005737, Year 2016 |
Publish date | Feb 10, 2016 (structure data deposition date) |
![]() | Lim, S.P. / Noble, C.G. / Seh, C.C. / Soh, T.S. / El Sahili, A. / Chan, G.K. / Lescar, J. / Arora, R. / Benson, T. / Nilar, S. ...Lim, S.P. / Noble, C.G. / Seh, C.C. / Soh, T.S. / El Sahili, A. / Chan, G.K. / Lescar, J. / Arora, R. / Benson, T. / Nilar, S. / Manjunatha, U. / Wan, K.F. / Dong, H. / Xie, X. / Shi, P.Y. / Yokokawa, F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.65 - 2.45 Å |
Structure data | ![]() PDB-5i3p: ![]() PDB-5i3q: ![]() PDB-5jjr: ![]() PDB-5jjs: ![]() PDB-5k5m: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-68T: ![]() ChemComp-HOH: ![]() ChemComp-68E: ![]() ChemComp-SAH: ![]() ChemComp-EDO: ![]() ChemComp-MG: ![]() ChemComp-PEG: ![]() ChemComp-6L2: ![]() ChemComp-MES: |
Source |
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![]() | TRANSFERASE/INHIBITOR / polymerase / dengue / TRANSFERASE-INHIBITOR complex / RdRP / HYDROLASE / RNA Dependent RNA Polymerase |