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-Structure paper
Title | Spectrum and Degree of CDK Drug Interactions Predicts Clinical Performance. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 15, Page 2273-2281, Year 2016 |
Publish date | Aug 1, 2016 (structure data deposition date) |
Authors | Chen, P. / Lee, N.V. / Hu, W. / Xu, M. / Ferre, R.A. / Lam, H. / Bergqvist, S. / Solowiej, J. / Diehl, W. / He, Y.A. ...Chen, P. / Lee, N.V. / Hu, W. / Xu, M. / Ferre, R.A. / Lam, H. / Bergqvist, S. / Solowiej, J. / Diehl, W. / He, Y.A. / Yu, X. / Nagata, A. / VanArsdale, T. / Murray, B.W. |
External links | Mol. Cancer Ther. / PubMed:27496135 |
Methods | X-ray diffraction |
Resolution | 2.27 - 2.8 Å |
Structure data | PDB-5l2i: PDB-5l2s: PDB-5l2t: PDB-5l2w: |
Chemicals | ChemComp-LQQ: ChemComp-6ZV: ChemComp-HOH: ChemComp-6ZZ: ChemComp-1QK: ChemComp-GOL: |
Source |
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Keywords | Transferase/Transferase Inhibitor / cyclin-dependent kinase / kinase inhibitor / kinase selectivity / Transferase-Transferase Inhibitor complex / Transferase/Cell Cycle/Inhibitor / Transferase-Cell Cycle-Inhibitor complex |