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-Structure paper
Title | Metabolic plasticity underpins innate and acquired resistance to LDHA inhibition. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 12, Page 779-786, Year 2016 |
Publish date | May 18, 2015 (structure data deposition date) |
![]() | Boudreau, A. / Purkey, H.E. / Hitz, A. / Robarge, K. / Peterson, D. / Labadie, S. / Kwong, M. / Hong, R. / Gao, M. / Del Nagro, C. ...Boudreau, A. / Purkey, H.E. / Hitz, A. / Robarge, K. / Peterson, D. / Labadie, S. / Kwong, M. / Hong, R. / Gao, M. / Del Nagro, C. / Pusapati, R. / Ma, S. / Salphati, L. / Pang, J. / Zhou, A. / Lai, T. / Li, Y. / Chen, Z. / Wei, B. / Yen, I. / Sideris, S. / McCleland, M. / Firestein, R. / Corson, L. / Vanderbilt, A. / Williams, S. / Daemen, A. / Belvin, M. / Eigenbrot, C. / Jackson, P.K. / Malek, S. / Hatzivassiliou, G. / Sampath, D. / Evangelista, M. / O'Brien, T. |
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Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-4zvv: |
Chemicals | ![]() ChemComp-NAD: ![]() ChemComp-SO4: ![]() ChemComp-GN0: ![]() ChemComp-HOH: |
Source |
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![]() | Oxidoreductase/Oxidoreductase Inhibitor / oxidoreductase inhibitor complex / LDHA-G02792140 / Oxidoreductase-Oxidoreductase Inhibitor complex |