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-Structure paper
Title | Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic Drugs. |
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Journal, issue, pages | J. Med. Chem., Vol. 59, Page 7598-7616, Year 2016 |
Publish date | Apr 15, 2016 (structure data deposition date) |
![]() | Borsari, C. / Luciani, R. / Pozzi, C. / Poehner, I. / Henrich, S. / Trande, M. / Cordeiro-da-Silva, A. / Santarem, N. / Baptista, C. / Tait, A. ...Borsari, C. / Luciani, R. / Pozzi, C. / Poehner, I. / Henrich, S. / Trande, M. / Cordeiro-da-Silva, A. / Santarem, N. / Baptista, C. / Tait, A. / Di Pisa, F. / Dello Iacono, L. / Landi, G. / Gul, S. / Wolf, M. / Kuzikov, M. / Ellinger, B. / Reinshagen, J. / Witt, G. / Gribbon, P. / Kohler, M. / Keminer, O. / Behrens, B. / Costantino, L. / Tejera Nevado, P. / Bifeld, E. / Eick, J. / Clos, J. / Torrado, J. / Jimenez-Anton, M.D. / Corral, M.J. / Alunda, J.M. / Pellati, F. / Wade, R.C. / Ferrari, S. / Mangani, S. / Costi, M.P. |
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Methods | X-ray diffraction |
Resolution | 1.38 - 1.78 Å |
Structure data | ![]() PDB-5jcj: ![]() PDB-5jcx: ![]() PDB-5jdc: ![]() PDB-5jdi: |
Chemicals | ![]() ChemComp-NAP: ![]() ChemComp-ACT: ![]() ChemComp-6JM: ![]() ChemComp-HOH: ![]() ChemComp-CC6: ![]() ChemComp-GOL: ![]() ChemComp-6JP: ![]() ChemComp-6JO: |
Source |
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![]() | OXIDOREDUCTASE / Trypanosoma brucei / pteridine reductase / oxydoreductase / inhibitor |