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-Structure paper
Title | Long-Range Inhibitor-Induced Conformational Regulation of Human IRE1 alpha Endoribonuclease Activity. |
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Journal, issue, pages | Mol. Pharmacol., Vol. 88, Page 1011-1023, Year 2015 |
Publish date | Mar 24, 2015 (structure data deposition date) |
Authors | Concha, N.O. / Smallwood, A. / Bonnette, W. / Totoritis, R. / Zhang, G. / Federowicz, K. / Yang, J. / Qi, H. / Chen, S. / Campobasso, N. ...Concha, N.O. / Smallwood, A. / Bonnette, W. / Totoritis, R. / Zhang, G. / Federowicz, K. / Yang, J. / Qi, H. / Chen, S. / Campobasso, N. / Choudhry, A.E. / Shuster, L.E. / Evans, K.A. / Ralph, J. / Sweitzer, S. / Heerding, D.A. / Buser, C.A. / Su, D.S. / DeYoung, M.P. |
External links | Mol. Pharmacol. / PubMed:26438213 |
Methods | X-ray diffraction |
Resolution | 2.463 - 3.102 Å |
Structure data | PDB-4yz9: PDB-4yzc: PDB-4yzd: |
Chemicals | ChemComp-4K7: ChemComp-HOH: ChemComp-STU: ChemComp-MG: ChemComp-ADP: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / active / inhibitor / complex / IRE1 / TRANSFERASE-TRANSFERASE INHIBITOR complex / staurosporine / TRANSFERASE / ADP |