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Title | 9H-Purine Scaffold Reveals Induced-Fit Pocket Plasticity of the BRD9 Bromodomain. |
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Journal, issue, pages | J. Med. Chem., Vol. 58, Page 2718-2736, Year 2015 |
Publish date | Feb 2, 2015 (structure data deposition date) |
![]() | Picaud, S. / Strocchia, M. / Terracciano, S. / Lauro, G. / Mendez, J. / Daniels, D.L. / Riccio, R. / Bifulco, G. / Bruno, I. / Filippakopoulos, P. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 2.05 Å |
Structure data | ![]() PDB-4xy8: ![]() PDB-4xy9: ![]() PDB-4xya: |
Chemicals | ![]() ChemComp-43U: ![]() ChemComp-BR: ![]() ChemComp-HOH: ![]() ChemComp-EDO: ![]() ChemComp-43S: |
Source |
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![]() | TRANSCRIPTION / Bromodomain / ligand / complex / Structural Genomics Consortium / SGC |