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-Structure paper
Title | Structure-Guided Design of a High Affinity Inhibitor to Human CtBP. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 10, Page 1118-1127, Year 2015 |
Publish date | Jul 29, 2014 (structure data deposition date) |
Authors | Hilbert, B.J. / Morris, B.L. / Ellis, K.C. / Paulsen, J.L. / Schiffer, C.A. / Grossman, S.R. / Royer, W.E. |
External links | Acs Chem. Biol. / PubMed:25636004 |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.3 Å |
Structure data | PDB-4u6q: PDB-4u6s: |
Chemicals | ChemComp-NAI: ChemComp-3CR: ChemComp-CA: ChemComp-FMT: ChemComp-HOH: ChemComp-NAD: ChemComp-PPY: |
Source |
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Keywords | OXIDOREDUCTASE / Rossman fold / transcription regulator / cancer / inhibitor / substrate |