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| Title | A cyclic peptidic serine protease inhibitor: increasing affinity by increasing peptide flexibility. |
|---|---|
| Journal, issue, pages | Plos One, Vol. 9, Page e115872-e115872, Year 2014 |
| Publish date | Nov 25, 2014 (structure data deposition date) |
Authors | Zhao, B. / Xu, P. / Jiang, L. / Paaske, B. / Kromann-Hansen, T. / Jensen, J.K. / Srensen, H.P. / Liu, Z. / Nielsen, J.T. / Christensen, A. ...Zhao, B. / Xu, P. / Jiang, L. / Paaske, B. / Kromann-Hansen, T. / Jensen, J.K. / Srensen, H.P. / Liu, Z. / Nielsen, J.T. / Christensen, A. / Hosseini, M. / Srensen, K.K. / Nielsen, N.C. / Jensen, K.J. / Huang, M. / Andreasen, P.A. |
External links | Plos One / PubMed:25545505 |
| Methods | X-ray diffraction |
| Resolution | 1.8 - 2.28 Å |
| Structure data | ![]() PDB-4x1n: ![]() PDB-4x1q: ![]() PDB-4x1r: ![]() PDB-4x1s: |
| Chemicals | ![]() ChemComp-MRZ: ![]() ChemComp-HOH: ![]() ChemComp-PL0: |
| Source |
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Keywords | HYDROLASE INHIBITOR/HYDROLASE / Serine protease / peptidic inhibitor / uPA / HYDROLASE INHIBITOR-HYDROLASE complex |
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homo sapiens (human)
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