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-Structure paper
Title | Design and Synthesis of High-Affinity Dimeric Inhibitors Targeting the Interactions between Gephyrin and Inhibitory Neurotransmitter Receptors. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 54, Page 490-494, Year 2015 |
Publish date | Aug 5, 2014 (structure data deposition date) |
![]() | Maric, H.M. / Kasaragod, V.B. / Haugaard-Kedstrom, L. / Hausrat, T.J. / Kneussel, M. / Schindelin, H. / Strmgaard, K. |
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Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | ![]() PDB-4u90: ![]() PDB-4u91: |
Chemicals | ![]() ChemComp-BU1: ![]() ChemComp-3F8: ![]() ChemComp-HOH: ![]() ChemComp-ACT: ![]() ChemComp-EDO: ![]() ChemComp-CA: ![]() ChemComp-3F7: |
Source |
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![]() | TRANSFER PROTEIN / STRUCTURAL PROTEIN / Inhibitory synapse / Scaffolding protein / GABA type A receptor / transferase / transfer protein - structural protein complex |