+Search query
-Structure paper
Title | Structure of the BRAF-MEK Complex Reveals a Kinase Activity Independent Role for BRAF in MAPK Signaling. |
---|---|
Journal, issue, pages | Cancer Cell, Vol. 26, Page 402-413, Year 2014 |
Publish date | Sep 10, 2013 (structure data deposition date) |
![]() | Haling, J.R. / Sudhamsu, J. / Yen, I. / Sideris, S. / Sandoval, W. / Phung, W. / Bravo, B.J. / Giannetti, A.M. / Peck, A. / Masselot, A. ...Haling, J.R. / Sudhamsu, J. / Yen, I. / Sideris, S. / Sandoval, W. / Phung, W. / Bravo, B.J. / Giannetti, A.M. / Peck, A. / Masselot, A. / Morales, T. / Smith, D. / Brandhuber, B.J. / Hymowitz, S.G. / Malek, S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.802 - 2.8483 Å |
Structure data | ![]() PDB-4mne: ![]() PDB-4mnf: |
Chemicals | ![]() ChemComp-ACP: ![]() ChemComp-MG: ![]() ChemComp-573: ![]() ChemComp-CL: ![]() ChemComp-HOH: ![]() ChemComp-29L: |
Source |
|
![]() | TRANSFERASE/TRANSFERASE INHIBITOR / RAF / MAPK / kinase domain / ATP-binding / ERK / RAS / PAK / TRANSFERASE-TRANSFERASE INHIBITOR complex / active conformation |