+Search query
-Structure paper
Title | PARP Inhibitor with Selectivity Toward ADP-Ribosyltransferase ARTD3/PARP3 |
---|---|
Journal, issue, pages | Acs Chem. Biol., Vol. 8, Page 1698-1703, Year 2013 |
Publish date | Aug 30, 2012 (structure data deposition date) |
Authors | Lindgren, A.E.G. / Karlberg, T. / Thorsell, A.G. / Hesse, M. / Spjut, S. / Ekblad, T. / Andersson, C.D. / Pinto, A.F. / Weigelt, J. / Hottiger, M.O. ...Lindgren, A.E.G. / Karlberg, T. / Thorsell, A.G. / Hesse, M. / Spjut, S. / Ekblad, T. / Andersson, C.D. / Pinto, A.F. / Weigelt, J. / Hottiger, M.O. / Linusson, A. / Elofsson, M. / Schuler, H. |
External links | Acs Chem. Biol. / PubMed:23742272 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.89 Å |
Structure data | PDB-4gv0: PDB-4gv2: PDB-4gv4: PDB-4gv7: |
Chemicals | ChemComp-8ME: ChemComp-DMS: ChemComp-HOH: ChemComp-5ME: ChemComp-MEJ: ChemComp-MEW: |
Source |
|
Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / NAD / ADP-RIBOSE / PARP3 / ARTD3 / ARTD TRANSFERASE DOMAIN / ADP-RIBOSYLATION / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX / TRANSFERASE / ADP- RIBOSYLATION / PARP1 / ARTD1 / ADP-RIBOSE TRANSFERASE |