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Title | Structural Basis and SAR for G007-LK, a Lead Stage 1,2,4-Triazole Based Specific Tankyrase 1/2 Inhibitor. |
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Journal, issue, pages | J. Med. Chem., Vol. 56, Page 3012-3023, Year 2013 |
Publish date | Nov 13, 2012 (structure data deposition date) |
Authors | Voronkov, A. / Holsworth, D.D. / Waaler, J. / Wilson, S.R. / Ekblad, B. / Perdreau-Dahl, H. / Dinh, H. / Drewes, G. / Hopf, C. / Morth, J.P. / Krauss, S. |
External links | J. Med. Chem. / PubMed:23473363 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-4hyf: |
Chemicals | ChemComp-NCA: ChemComp-ZN: ChemComp-1AK: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / CATALYTIC FRAGMENT / PARP / ADP-RIBOSYLATION / ANK REPEAT / CHROMOSOMAL PROTEIN / GLYCOSYLTRANSFERASE / PHOSPHORYLATION / TELOMERE / TRANSFERASE / TRANSLOCATION / TRANSPORT / WNT-SIGNALLING / TRANSFERASE-TRANSFERASE INHIBITOR complex |