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-Structure paper
Title | Identification of Cys255 in HIF-1 alpha as a novel site for development of covalent inhibitors of HIF-1 alpha /ARNT PasB domain protein-protein interaction. |
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Journal, issue, pages | Protein Sci., Vol. 21, Page 1885-1896, Year 2012 |
Publish date | Sep 19, 2012 (structure data deposition date) |
![]() | Cardoso, R. / Love, R. / Nilsson, C.L. / Bergqvist, S. / Nowlin, D. / Yan, J. / Liu, K.K. / Zhu, J. / Chen, P. / Deng, Y.L. ...Cardoso, R. / Love, R. / Nilsson, C.L. / Bergqvist, S. / Nowlin, D. / Yan, J. / Liu, K.K. / Zhu, J. / Chen, P. / Deng, Y.L. / Dyson, H.J. / Greig, M.J. / Brooun, A. |
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Methods | X-ray diffraction |
Resolution | 1.52 Å |
Structure data | ![]() PDB-4h6j: |
Chemicals | ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / PAS DOMAIN / HETERODIMER / HYPOXIA INDUCIBLE FACTOR / TRANSCRIPTION FACTOR / ARNT |