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-Structure paper
Title | Fragment based discovery of a novel and selective PI3 kinase inhibitor. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 21, Page 6586-6590, Year 2011 |
Publish date | Jul 27, 2011 (structure data deposition date) |
Authors | Hughes, S.J. / Millan, D.S. / Kilty, I.C. / Lewthwaite, R.A. / Mathias, J.P. / O'Reilly, M.A. / Pannifer, A. / Phelan, A. / Stuhmeier, F. / Baldock, D.A. / Brown, D.G. |
External links | Bioorg. Med. Chem. Lett. / PubMed:21925880 |
Methods | X-ray diffraction |
Resolution | 2.5 - 2.8 Å |
Structure data | PDB-3zvv: PDB-3zw3: |
Chemicals | ChemComp-XAZ: ChemComp-HOH: ChemComp-ZW3: |
Source |
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Keywords | TRANSFERASE / PI3 KINASE GAMMA |