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TitleDiscovery of the first non-ATP competitive IGF-1R kinase inhibitors: Advantages in comparison with competitive inhibitors
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 21, Page 2224-2228, Year 2011
Publish dateJul 22, 2010 (structure data deposition date)
AuthorsLesuisse, D. / Mauger, J. / Nemecek, C. / Maignan, S. / Boiziau, J. / Harlow, G. / Hittinger, A. / Ruf, S. / Strobel, H. / Nair, A. ...Lesuisse, D. / Mauger, J. / Nemecek, C. / Maignan, S. / Boiziau, J. / Harlow, G. / Hittinger, A. / Ruf, S. / Strobel, H. / Nair, A. / Ritter, K. / Malleron, J.L. / Dagallier, A. / El-Ahmad, Y. / Guilloteau, J.P. / Guizani, H. / Bouchard, H. / Venot, C.
External linksBioorg. Med. Chem. Lett. / PubMed:21441024
MethodsX-ray diffraction
Resolution2.1 Å
Structure data

PDB-3o23:
Human unphosphorylated IGF1-R Kinase domain in complex with an hydantoin inhibitor
Method: X-RAY DIFFRACTION / Resolution: 2.1 Å

Chemicals

ChemComp-MQY:
(5S)-5-methyl-1-(quinolin-4-ylmethyl)-3-{4-[(trifluoromethyl)sulfonyl]phenyl}imidazolidine-2,4-dione

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsTRANSFERASE/TRANSFERASE INHIBITOR / Protein Kinase / TRANSFERASE-TRANSFERASE INHIBITOR complex

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