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-Structure paper
Title | Selective inhibition of BET bromodomains. |
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Journal, issue, pages | Nature, Vol. 468, Page 1067-1073, Year 2010 |
Publish date | May 7, 2010 (structure data deposition date) |
![]() | Filippakopoulos, P. / Qi, J. / Picaud, S. / Shen, Y. / Smith, W.B. / Fedorov, O. / Morse, E.M. / Keates, T. / Hickman, T.T. / Felletar, I. ...Filippakopoulos, P. / Qi, J. / Picaud, S. / Shen, Y. / Smith, W.B. / Fedorov, O. / Morse, E.M. / Keates, T. / Hickman, T.T. / Felletar, I. / Philpott, M. / Munro, S. / McKeown, M.R. / Wang, Y. / Christie, A.L. / West, N. / Cameron, M.J. / Schwartz, B. / Heightman, T.D. / La Thangue, N. / French, C.A. / Wiest, O. / Kung, A.L. / Knapp, S. / Bradner, J.E. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 1.61 Å |
Structure data | ![]() PDB-3mxf: ![]() PDB-3oni: |
Chemicals | ![]() ChemComp-JQ1: ![]() ChemComp-IOD: ![]() ChemComp-EDO: ![]() ChemComp-DMS: ![]() ChemComp-HOH: ![]() ChemComp-NI: |
Source |
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![]() | CELL CYCLE / Bromodomain-containing protein 4 isoform long / BRD4 / Bromodomain containing protein 4 / CAP / HUNK1 / MCAP / Mitotic chromosome associated protein / JQ1 / betsoff1 / Structural Genomics Consortium / SGC / Structural Genomics / Bromodomain / Inhibition / Probe |