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| Title | Structural basis for binding of cyclic 2-oxoglutarate analogues to factor-inhibiting hypoxia-inducible factor. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 20, Page 6125-6128, Year 2010 |
| Publish date | Oct 10, 2008 (structure data deposition date) |
Authors | Conejo-Garcia, A. / McDonough, M.A. / Loenarz, C. / McNeill, L.A. / Hewitson, K.S. / Ge, W. / Lienard, B.M. / Schofield, C.J. / Clifton, I.J. |
External links | Bioorg. Med. Chem. Lett. / PubMed:20822901 |
| Methods | X-ray diffraction |
| Resolution | 2.12 - 2.5 Å |
| Structure data | ![]() PDB-2w0x: ![]() PDB-2wa3: ![]() PDB-2wa4: |
| Chemicals | ![]() ChemComp-FE2: ![]() ChemComp-PD2: ![]() ChemComp-SO4: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-A29: ![]() ChemComp-069: |
| Source |
|
Keywords | OXIDOREDUCTASE / HYDROXYLASE / DIOXYGENASE / TRANSCRIPTION / TRANSCRIPTION ACTIVATOR/INHIBITOR / HYPOXIA |
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homo sapiens (human)
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