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-Structure paper
Title | Design of selective, ATP-competitive inhibitors of Akt. |
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Journal, issue, pages | J. Med. Chem., Vol. 53, Page 4615-4622, Year 2010 |
Publish date | May 3, 2010 (structure data deposition date) |
![]() | Freeman-Cook, K.D. / Autry, C. / Borzillo, G. / Gordon, D. / Barbacci-Tobin, E. / Bernardo, V. / Briere, D. / Clark, T. / Corbett, M. / Jakubczak, J. ...Freeman-Cook, K.D. / Autry, C. / Borzillo, G. / Gordon, D. / Barbacci-Tobin, E. / Bernardo, V. / Briere, D. / Clark, T. / Corbett, M. / Jakubczak, J. / Kakar, S. / Knauth, E. / Lippa, B. / Luzzio, M.J. / Mansour, M. / Martinelli, G. / Marx, M. / Nelson, K. / Pandit, J. / Rajamohan, F. / Robinson, S. / Subramanyam, C. / Wei, L. / Wythes, M. / Morris, J. |
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Methods | X-ray diffraction |
Resolution | 2.01 - 2.49 Å |
Structure data | ![]() PDB-3mv5: ![]() PDB-3mvh: ![]() PDB-3mvj: |
Chemicals | ![]() ChemComp-MN: ![]() ChemComp-XFE: ![]() ChemComp-HOH: ![]() ChemComp-WFE: |
Source |
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![]() | TRANSFERASE / kinase inhibitor |