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-Structure paper
Title | Structural and mechanistic basis for a new mode of glycosyltransferase inhibition. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 6, Page 321-323, Year 2010 |
Publish date | Aug 14, 2009 (structure data deposition date) |
![]() | Pesnot, T. / Jorgensen, R. / Palcic, M.M. / Wagner, G.K. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.25 - 1.651 Å |
Structure data | ![]() PDB-3ioh: ![]() PDB-3ioi: ![]() PDB-3ioj: |
Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-MN: ![]() ChemComp-SO4: ![]() ChemComp-1GW: ![]() ChemComp-UDP: |
Source |
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![]() | TRANSFERASE / GTA / ABO / cisAB mutant / AA(Gly)B / ROSSMANN FOLD / UNLIGANDED / OPEN CONFORMATION / BLOOD GROUP ANTIGEN / GLYCOPROTEIN / GLYCOSYLTRANSFERASE / GOLGI APPARATUS / MANGANESE / MEMBRANE / METAL-BINDING / POLYMORPHISM / SECRETED / SIGNAL-ANCHOR / TRANSMEMBRANE / INHIBITOR / SEMI-CLOSED CONFORMATION / UDP |