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Structure paper

TitleX-ray crystallographic analysis of alpha-ketoheterocycle inhibitors bound to a humanized variant of fatty acid amide hydrolase.
Journal, issue, pagesJ. Med. Chem., Vol. 53, Page 230-240, Year 2010
Publish dateOct 13, 2009 (structure data deposition date)
AuthorsMileni, M. / Garfunkle, J. / Ezzili, C. / Kimball, F.S. / Cravatt, B.F. / Stevens, R.C. / Boger, D.L.
External linksJ. Med. Chem. / PubMed:19924997
MethodsX-ray diffraction
Resolution1.95 - 2.251 Å
Structure data

PDB-3k7f:
Crystal Structure Analysis of a Phenhexyl/Oxazole/Carboxypyridine alpha-Ketoheterocycle Inhibitor Bound to a Humanized Variant of Fatty Acid Amide Hydrolase'
Method: X-RAY DIFFRACTION / Resolution: 1.95 Å

PDB-3k83:
Crystal Structure Analysis of a Biphenyl/Oxazole/Carboxypyridine alpha-ketoheterocycle Inhibitor Bound to a Humanized Variant of Fatty Acid Amide Hydrolase
Method: X-RAY DIFFRACTION / Resolution: 2.251 Å

PDB-3k84:
Crystal Structure Analysis of a Oleyl/Oxadiazole/pyridine Inhibitor Bound to a Humanized Variant of Fatty Acid Amide Hydrolase
Method: X-RAY DIFFRACTION / Resolution: 2.25 Å

Chemicals

ChemComp-F2C:
6-[2-(7-phenylheptanoyl)-1,3-oxazol-5-yl]pyridine-2-carboxylic acid

ChemComp-CL:
Unknown entry

ChemComp-NA:
Unknown entry

ChemComp-HOH:
WATER

ChemComp-F27:
6-[2-(3-biphenyl-4-ylpropanoyl)-1,3-oxazol-5-yl]pyridine-2-carboxylic acid

ChemComp-1DO:
1-DODECANOL

ChemComp-K84:
(9Z)-1-(5-pyridin-2-yl-1,3,4-oxadiazol-2-yl)octadec-9-en-1-one

Source
  • rattus norvegicus (Norway rat)
KeywordsHYDROLASE / protein-inhibitor complex / FAAH / oxazole / Membrane / Transmembrane / conjugate / covalent modification / monotopic / fatty acid / serine hydrolase / endocannabinoid / reversible inhibitor. / oxadiazole / alpha-ketoheterocycle

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