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Title | Discovery and design of novel HSP90 inhibitors using multiple fragment-based design strategies. |
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Journal, issue, pages | Chem. Biol. Drug Des., Vol. 70, Page 1-12, Year 2007 |
Publish date | Jun 26, 2007 (structure data deposition date) |
![]() | Huth, J.R. / Park, C. / Petros, A.M. / Kunzer, A.R. / Wendt, M.D. / Wang, X. / Lynch, C.L. / Mack, J.C. / Swift, K.M. / Judge, R.A. ...Huth, J.R. / Park, C. / Petros, A.M. / Kunzer, A.R. / Wendt, M.D. / Wang, X. / Lynch, C.L. / Mack, J.C. / Swift, K.M. / Judge, R.A. / Chen, J. / Richardson, P.L. / Jin, S. / Tahir, S.K. / Matayoshi, E.D. / Dorwin, S.A. / Ladror, U.S. / Severin, J.M. / Walter, K.A. / Bartley, D.M. / Fesik, S.W. / Elmore, S.W. / Hajduk, P.J. |
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Methods | X-ray diffraction |
Resolution | 1.68 - 3.1 Å |
Structure data | ![]() PDB-2qf6: ![]() PDB-2qfo: ![]() PDB-2qg0: ![]() PDB-2qg2: |
Chemicals | ![]() ChemComp-A56: ![]() ChemComp-HOH: ![]() ChemComp-A13: ![]() ChemComp-A51: ![]() ChemComp-A94: ![]() ChemComp-A91: |
Source |
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