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-Structure paper
Title | Discovery and characterization of a novel inhibitor of matrix metalloprotease-13 that reduces cartilage damage in vivo without joint fibroplasia side effects. |
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Journal, issue, pages | J. Biol. Chem., Vol. 282, Page 27781-27791, Year 2007 |
Publish date | Feb 15, 2007 (structure data deposition date) |
![]() | Johnson, A.R. / Pavlovsky, A.G. / Ortwine, D.F. / Prior, F. / Man, C.F. / Bornemeier, D.A. / Banotai, C.A. / Mueller, W.T. / McConnell, P. / Yan, C. ...Johnson, A.R. / Pavlovsky, A.G. / Ortwine, D.F. / Prior, F. / Man, C.F. / Bornemeier, D.A. / Banotai, C.A. / Mueller, W.T. / McConnell, P. / Yan, C. / Baragi, V. / Lesch, C. / Roark, W.H. / Wilson, M. / Datta, K. / Guzman, R. / Han, H.K. / Dyer, R.D. |
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Methods | X-ray diffraction |
Resolution | 1.74 - 2.3 Å |
Structure data | ![]() PDB-2ow9: ![]() PDB-2ozr: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-CA: ![]() ChemComp-SO4: ![]() ChemComp-SP6: ![]() ChemComp-HAE: ![]() ChemComp-HOH: ![]() ChemComp-GG1: |
Source |
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![]() | HYDROLASE / Complex crystal structure / Martix Metalloproteinase / MMP13 / Specific MMP13 inhibitor / S1' MMP13 inhibitor / Crystal Complex Structure / Matrix Metalloproteinase / MMP13 Catalytic Domain / MMP13 Specific Inhibitor |