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-Structure paper
Title | Structure-guided design of Peptide-based tryptase inhibitors. |
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Journal, issue, pages | Biochemistry, Vol. 45, Page 5964-5973, Year 2006 |
Publish date | Jan 17, 2006 (structure data deposition date) |
Authors | McGrath, M.E. / Sprengeler, P.A. / Hirschbein, B. / Somoza, J.R. / Lehoux, I. / Janc, J.W. / Gjerstad, E. / Graupe, M. / Estiarte, A. / Venkataramani, C. ...McGrath, M.E. / Sprengeler, P.A. / Hirschbein, B. / Somoza, J.R. / Lehoux, I. / Janc, J.W. / Gjerstad, E. / Graupe, M. / Estiarte, A. / Venkataramani, C. / Liu, Y. / Yee, R. / Ho, J.D. / Green, M.J. / Lee, C.-S. / Liu, L. / Tai, V. / Spencer, J. / Sperandio, D. / Katz, B.A. |
External links | Biochemistry / PubMed:16681368 |
Methods | X-ray diffraction |
Resolution | 1.57 - 2.5 Å |
Structure data | PDB-2fpz: PDB-2fs8: PDB-2fs9: PDB-2fww: PDB-2fx4: PDB-2fx6: PDB-2fxr: |
Chemicals | ChemComp-270: ChemComp-HOH: ChemComp-C3A: ChemComp-C4A: ChemComp-C1R: ChemComp-CA: |
Source |
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Keywords | HYDROLASE / Serine protease / drug design / proteinase / 29382 / serine proteinase / 28427 / acylenzyme complex / fragment screening / S1 site / activated ketone inhibitor / pyrrolidine / CRA-29382 |