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-Structure paper
Title | Enhanced FTase activity achieved via piperazine interaction with catalytic zinc. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 16, Page 984-988, Year 2006 |
Publish date | Oct 24, 2005 (structure data deposition date) |
Authors | Njoroge, F.G. / Vibulbhan, B. / Pinto, P. / Strickland, C. / Bishop, W.R. / Nomeir, A. / Girijavallabhan, V. |
External links | Bioorg. Med. Chem. Lett. / PubMed:16298128 |
Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | PDB-2bed: |
Chemicals | ChemComp-ZN: ChemComp-FPP: ChemComp-736: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / FPT / PTase / Farnesyl / drug design |