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TitleStructure based approach to the design of bicyclic-1H-isoindole-1,3(2H)-dione based androgen receptor antagonists.
Journal, issue, pagesBioorg. Med. Chem. Lett., Vol. 15, Page 271-276, Year 2005
Publish dateOct 5, 2004 (structure data deposition date)
AuthorsSalvati, M.E. / Balog, A. / Shan, W. / Wei, D.D. / Pickering, D. / Attar, R.M. / Geng, J. / Rizzo, C.A. / Gottardis, M.M. / Weinmann, R. ...Salvati, M.E. / Balog, A. / Shan, W. / Wei, D.D. / Pickering, D. / Attar, R.M. / Geng, J. / Rizzo, C.A. / Gottardis, M.M. / Weinmann, R. / Krystek, S.R. / Sack, J. / An, Y. / Kish, K.
External linksBioorg. Med. Chem. Lett. / PubMed:15603938
MethodsX-ray diffraction
Resolution2.2 Å
Structure data

PDB-1xnn:
CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN T877A MUTANT COMPLEX WITH (3A-ALPHA-,4-ALPHA 7-ALPHA-,7A-ALPHA-)-3A,4,7,7A-TETRAHYDRO-2-(4-NITRO-1-NAPHTHALENYL)-4,7-ETHANO-1H-ISOINDOLE-1,3(2H)-DIONE.
Method: X-RAY DIFFRACTION / Resolution: 2.2 Å

Chemicals

ChemComp-HYQ:
REL-(3AR,4S,7R,7AS)-3A,4,7,7A-TETRAHYDRO-2-(4-NITRO-1-NAPHTHALENYL)-4,7-ETHANO-1H-ISOINDOLE-1,3(2H)-DIONE

ChemComp-HOH:
WATER

Source
  • rattus norvegicus (Norway rat)
KeywordsHORMONE/GROWTH FACTOR / ANDROGEN RECEPTOR / STEROID RECEPTOR / NUCLEAR RECEPTOR / TRANSCRIPTION REGULATION / LIGAND-BINDING DOMAIN / HORMONE-GROWTH FACTOR COMPLEX

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