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-Structure paper
Title | Structural Basis for Ucn-01 (7-Hydroxystaurosporine) Specificity and Pdk1 (3-Phosphoinositide-Dependent Protein Kinase-1) Inhibition |
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Journal, issue, pages | Biochem. J., Vol. 375, Page 255-, Year 2003 |
Publish date | Aug 1, 2003 (structure data deposition date) |
![]() | Komander, D. / Kular, G.S. / Bain, J. / Elliot, M. / Alessi, D.R. / Van Aalten, D.M.F. |
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Methods | X-ray diffraction |
Resolution | 2.3 - 2.51 Å |
Structure data | ![]() PDB-1oky: ![]() PDB-1okz: |
Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-STU: ![]() ChemComp-HOH: ![]() ChemComp-UCN: |
Source |
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![]() | TRANSFERASE / PROTEIN KINASE / PKB / PDK1 / STAUROSPORINE / UCN-01 / 7-HYDROXY STAUROSPORINE / INHIBITOR / ATP-BINDING / PHOSPHORYLATION |