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| Title | Catalytically active MAP KAP kinase 2 structures in complex with staurosporine and ADP reveal differences with the autoinhibited enzyme |
|---|---|
| Journal, issue, pages | Structure, Vol. 11, Page 627-636, Year 2003 |
| Publish date | Feb 10, 2003 (structure data deposition date) |
Authors | Underwood, K.W. / Parris, K.D. / Federico, E. / Mosyak, L. / Czerwinski, R.M. / Shane, T. / Taylor, M. / Svenson, K. / Liu, Y. / Hsiao, C.L. ...Underwood, K.W. / Parris, K.D. / Federico, E. / Mosyak, L. / Czerwinski, R.M. / Shane, T. / Taylor, M. / Svenson, K. / Liu, Y. / Hsiao, C.L. / Wolfrom, S. / Maguire, M. / Malakian, K. / Telliez, J.B. / Lin, L.L. / Kriz, R.W. / Seehra, J. / Somers, W.S. / Stahl, M.L. |
External links | Structure / PubMed:12791252 |
| Methods | X-ray diffraction |
| Resolution | 2.7 - 3 Å |
| Structure data | ![]() PDB-1nxk: ![]() PDB-1ny3: |
| Chemicals | ![]() ChemComp-STU: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-ADP: |
| Source |
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Keywords | TRANSFERASE / protein kinase / mk2 / phosphorylation / staurosporine / MAP KAP kinase 2 / ADP / kinase / ser/thr kinase |
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homo sapiens (human)
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