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Title | Binding of N-acetyl-N '-beta-D-glucopyranosyl urea and N-benzoyl-N '-beta-D-glucopyranosyl urea to glycogen phosphorylase b: kinetic and crystallographic studies. |
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Journal, issue, pages | Eur. J. Biochem., Vol. 269, Page 1684-1696, Year 2002 |
Publish date | Sep 18, 2001 (structure data deposition date) |
Authors | Oikonomakos, N.G. / Kosmopoulou, M. / Zographos, S.E. / Leonidas, D.D. / Chrysina, E.D. / Somsak, L. / Nagy, V. / Praly, J.P. / Docsa, T. / Toth, B. / Gergely, P. |
External links | Eur. J. Biochem. / PubMed:11895439 |
Methods | X-ray diffraction |
Resolution | 1.8 - 2.26 Å |
Structure data | PDB-1k06: PDB-1k08: PDB-1kti: |
Chemicals | ChemComp-BZD: ChemComp-PLP: ChemComp-HOH: ChemComp-AZC: |
Source |
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Keywords | TRANSFERASE / glycogen phosphorylase / catalytic site / new allosteric site / GLYCOGENOLYSIS / TYPE 2 DIABETES |