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-Structure paper
Title | Structural mechanism for STI-571 inhibition of abelson tyrosine kinase. |
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Journal, issue, pages | Science, Vol. 289, Page 1938-1942, Year 2000 |
Publish date | Aug 31, 2000 (structure data deposition date) |
Authors | Schindler, T. / Bornmann, W. / Pellicena, P. / Miller, W.T. / Clarkson, B. / Kuriyan, J. |
External links | Science / PubMed:10988075 |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | PDB-1fpu: |
Chemicals | ChemComp-PRC: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / kinase / kinase inhibitor / STI-571 / activation loop |