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-Structure paper
Title | Lamivudine (3TC) resistance in HIV-1 reverse transcriptase involves steric hindrance with beta-branched amino acids. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 96, Page 10027-10032, Year 1999 |
Publish date | May 24, 2002 (structure data deposition date) |
Authors | Sarafianos, S.G. / Das, K. / Clark Jr., A.D. / Ding, J. / Boyer, P.L. / Hughes, S.H. / Arnold, E. |
External links | Proc. Natl. Acad. Sci. USA / PubMed:10468556 |
Methods | X-ray diffraction |
Resolution | 2.85 - 3.5 Å |
Structure data | PDB-1j5o: PDB-1qe1: |
Source |
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Keywords | TRANSFERASE/IMMUNE SYSTEM/DNA / HIV / REVERSE TRANSCRIPTASE / MET184ILE / 3TC / PROTEIN-DNA COMPLEX / DRUG RESISTANCE / M184I / TRANSFERASE-IMMUNE SYSTEM-DNA COMPLEX / TRANSFERASE / RESISTANCE / MUTANT / DNA POLYMERASE |