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-Structure paper
Title | Structure of acetylcholinesterase complexed with E2020 (Aricept): implications for the design of new anti-Alzheimer drugs. |
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Journal, issue, pages | Structure Fold. Des., Vol. 7, Page 297-307, Year 1999 |
Publish date | Mar 4, 1998 (structure data deposition date) |
Authors | Kryger, G. / Silman, I. / Sussman, J.L. |
External links | Structure Fold. Des. / PubMed:10368299 |
Methods | X-ray diffraction |
Resolution | 2.5 Å |
Structure data | PDB-1eve: |
Chemicals | ChemComp-NAG: ChemComp-E20: ChemComp-HOH: |
Source |
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Keywords | SERINE HYDROLASE / ALZHEIMER'S DISEASE / DRUG / ALPHA/BETA HYDROLASE / NEUROTRANSMITTER CLEAVAGE / CATALYTIC TRIAD / GLYCOSYLATED PROTEIN |