登録情報 データベース : PDB / ID : 8q6h 構造の表示 ダウンロードとリンクタイトル HUMAN PI4KIIIB IN COMPLEX WITH COVALENTLY BOUND INHIBITOR (COMPOUND 11) 要素Phosphatidylinositol 4-kinase beta 詳細 キーワード TRANSFERASE (転移酵素) / LIPID KINASE (キナーゼ) / TRANSFERASE-SIGNALING PROTEIN COMPLEX / COVALENT INHIBITOR.機能・相同性 機能・相同性情報分子機能 ドメイン・相同性 構成要素
1-phosphatidylinositol 4-kinase / 1-phosphatidylinositol 4-kinase activity / rough endoplasmic reticulum membrane / Synthesis of PIPs at the Golgi membrane / phosphatidylinositol biosynthetic process / phosphatidylinositol-mediated signaling / lysosome organization / inner ear development / phosphatidylinositol phosphate biosynthetic process / receptor-mediated endocytosis ... 1-phosphatidylinositol 4-kinase / 1-phosphatidylinositol 4-kinase activity / rough endoplasmic reticulum membrane / Synthesis of PIPs at the Golgi membrane / phosphatidylinositol biosynthetic process / phosphatidylinositol-mediated signaling / lysosome organization / inner ear development / phosphatidylinositol phosphate biosynthetic process / receptor-mediated endocytosis / 14-3-3 protein binding / kinase activity / mitochondrial outer membrane / エンドソーム / リン酸化 / ゴルジ体 / perinuclear region of cytoplasm / ゴルジ体 / シグナル伝達 / ATP binding / 生体膜 / 細胞質基質 / 細胞質 類似検索 - 分子機能 : / PI4KB/PIK1, accessory (PIK) domain / Phosphoinositide 3-kinase, accessory (PIK) domain / Phosphatidylinositol kinase / PIK helical domain profile. / Phosphatidylinositol 3- and 4-kinases signature 1. / Phosphatidylinositol 3/4-kinase, conserved site / Phosphatidylinositol 3- and 4-kinases signature 2. / Phosphatidylinositol 3-/4-kinase, catalytic domain superfamily / Phosphoinositide 3-kinase, catalytic domain ... : / PI4KB/PIK1, accessory (PIK) domain / Phosphoinositide 3-kinase, accessory (PIK) domain / Phosphatidylinositol kinase / PIK helical domain profile. / Phosphatidylinositol 3- and 4-kinases signature 1. / Phosphatidylinositol 3/4-kinase, conserved site / Phosphatidylinositol 3- and 4-kinases signature 2. / Phosphatidylinositol 3-/4-kinase, catalytic domain superfamily / Phosphoinositide 3-kinase, catalytic domain / Phosphatidylinositol 3- and 4-kinase / Phosphatidylinositol 3- and 4-kinases catalytic domain profile. / Phosphatidylinositol 3-/4-kinase, catalytic domain / Protein kinase-like domain superfamily 類似検索 - ドメイン・相同性 Chem-KI7 / Phosphatidylinositol 4-kinase beta / Phosphatidylinositol 4-kinase beta 類似検索 - 構成要素生物種 Homo sapiens (ヒト)手法 X線回折 / シンクロトロン / フーリエ合成 / 解像度 : 1.94 Å 詳細データ登録者 Somers, D.O. 資金援助 1件 詳細 詳細を隠す 引用ジャーナル : Rsc Chem Biol / 年 : 2023タイトル : Covalent targeting of non-cysteine residues in PI4KIII beta.著者 : Cosgrove, B. / Grant, E.K. / Bertrand, S. / Down, K.D. / Somers, D.O. / P Evans, J. / Tomkinson, N.C.O. / Barker, M.D. 履歴 登録 2023年8月11日 登録サイト : PDBE / 処理サイト : PDBE改定 1.0 2023年12月13日 Provider : repository / タイプ : Initial release