登録情報 | データベース: PDB / ID: 8wdx |
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タイトル | Crystal structure of human FABP4 complexed with C3 |
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要素 | Fatty acid-binding protein, adipocyte |
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キーワード | LIPID BINDING PROTEIN/INHIBITOR / lipid binding protein-inhibitor complex |
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機能・相同性 | 機能・相同性情報
hormone receptor binding / long-chain fatty acid transmembrane transporter activity / cellular response to lithium ion / long-chain fatty acid binding / Triglyceride catabolism / white fat cell differentiation / long-chain fatty acid transport / brown fat cell differentiation / fatty acid transport / lipid droplet ...hormone receptor binding / long-chain fatty acid transmembrane transporter activity / cellular response to lithium ion / long-chain fatty acid binding / Triglyceride catabolism / white fat cell differentiation / long-chain fatty acid transport / brown fat cell differentiation / fatty acid transport / lipid droplet / cholesterol homeostasis / fatty acid binding / response to bacterium / Transcriptional regulation of white adipocyte differentiation / positive regulation of inflammatory response / positive regulation of cold-induced thermogenesis / cellular response to tumor necrosis factor / negative regulation of DNA-templated transcription / extracellular exosome / nucleus / cytosol / cytoplasm類似検索 - 分子機能 Cytosolic fatty-acid binding proteins signature. / Intracellular lipid binding protein / Cytosolic fatty-acid binding / Lipocalin/cytosolic fatty-acid binding domain / Lipocalin / cytosolic fatty-acid binding protein family / Calycin類似検索 - ドメイン・相同性 Chem-W6K / Fatty acid-binding protein, adipocyte類似検索 - 構成要素 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 1.65 Å |
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データ登録者 | Xie, H. / Chen, G.F. / Xu, Y.C. |
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資金援助 | 1件 |
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引用 | ジャーナル: Eur.J.Med.Chem. / 年: 2023 タイトル: Structure-based design of potent FABP4 inhibitors with high selectivity against FABP3. 著者: Chen, G. / Xie, H. / You, M. / Liu, J. / Shao, Q. / Li, M. / Su, H. / Xu, Y. |
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履歴 | 登録 | 2023年9月16日 | 登録サイト: PDBJ / 処理サイト: PDBJ |
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改定 1.0 | 2023年12月27日 | Provider: repository / タイプ: Initial release |
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