登録情報 | データベース: PDB / ID: 8qvk |
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タイトル | Comparison of room-temperature and cryogenic structures of soluble Epoxide Hydrolase with ligands bound. |
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要素 | Bifunctional epoxide hydrolase 2 |
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キーワード | HYDROLASE / Inhibitor / serial crystallography / drug discovery / fixed target / room temperature / microcrystals |
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機能・相同性 | 機能・相同性情報
lipid-phosphate phosphatase / 10-hydroxy-9-(phosphonooxy)octadecanoate phosphatase activity / stilbene catabolic process / phospholipid dephosphorylation / lipid phosphatase activity / Biosynthesis of maresins / soluble epoxide hydrolase / epoxide metabolic process / lysophosphatidic acid phosphatase activity / Synthesis of epoxy (EET) and dihydroxyeicosatrienoic acids (DHET) ...lipid-phosphate phosphatase / 10-hydroxy-9-(phosphonooxy)octadecanoate phosphatase activity / stilbene catabolic process / phospholipid dephosphorylation / lipid phosphatase activity / Biosynthesis of maresins / soluble epoxide hydrolase / epoxide metabolic process / lysophosphatidic acid phosphatase activity / Synthesis of epoxy (EET) and dihydroxyeicosatrienoic acids (DHET) / epoxide hydrolase activity / regulation of cholesterol metabolic process / dephosphorylation / phosphatase activity / peroxisomal matrix / toxic substance binding / cholesterol homeostasis / Peroxisomal protein import / response to toxic substance / peroxisome / positive regulation of gene expression / magnesium ion binding / protein homodimerization activity / extracellular exosome / cytosol類似検索 - 分子機能 Predicted HAD-superfamily phosphatase, subfamily IA/Epoxide hydrolase, N-terminal / Phosphoglycolate phosphatase-like, domain 2 / HAD hydrolase, subfamily IA / Epoxide hydrolase-like / alpha/beta hydrolase fold / haloacid dehalogenase-like hydrolase / Alpha/beta hydrolase fold-1 / HAD superfamily / HAD-like superfamily / Alpha/Beta hydrolase fold類似検索 - ドメイン・相同性 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 2.1 Å |
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データ登録者 | Dunge, A. / Uwangue, O. / Phan, C. / Bjelcic, M. / Gunnarsson, J. / Wehlander, G. / Kack, H. / Branden, G. |
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資金援助 | スウェーデン, 4件 組織 | 認可番号 | 国 |
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The Swedish Foundation for Strategic Research | ID17-0060 | スウェーデン | Swedish Research Council | 2017-06734 | スウェーデン | Swedish Research Council | 2021-05662 | スウェーデン | Swedish Research Council | 2021-05981 | スウェーデン |
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引用 | ジャーナル: Iucrj / 年: 2024 タイトル: Exploring serial crystallography for drug discovery. 著者: Dunge, A. / Phan, C. / Uwangue, O. / Bjelcic, M. / Gunnarsson, J. / Wehlander, G. / Kack, H. / Branden, G. |
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履歴 | 登録 | 2023年10月18日 | 登録サイト: PDBE / 処理サイト: PDBE |
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改定 1.0 | 2024年8月14日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2024年9月11日 | Group: Database references / カテゴリ: citation / citation_author Item: _citation.journal_volume / _citation.page_first ..._citation.journal_volume / _citation.page_first / _citation.page_last / _citation_author.identifier_ORCID |
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