- PDB-7qhw: TTBK1 kinase domain in complex with inhibitor 29 -
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IDまたはキーワード:
読み込み中...
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基本情報
登録情報
データベース: PDB / ID: 7qhw
タイトル
TTBK1 kinase domain in complex with inhibitor 29
要素
Tau-tubulin kinase 1
キーワード
TRANSFERASE / kinase / inhibitor
機能・相同性
機能・相同性情報
positive regulation of cyclin-dependent protein kinase activity / positive regulation of astrocyte activation / positive regulation of microglial cell activation / positive regulation of cysteine-type endopeptidase activity / microtubule associated complex / positive regulation of protein polymerization / tau-protein kinase activity / substantia nigra development / negative regulation of protein binding / peptidyl-threonine phosphorylation ...positive regulation of cyclin-dependent protein kinase activity / positive regulation of astrocyte activation / positive regulation of microglial cell activation / positive regulation of cysteine-type endopeptidase activity / microtubule associated complex / positive regulation of protein polymerization / tau-protein kinase activity / substantia nigra development / negative regulation of protein binding / peptidyl-threonine phosphorylation / tau protein binding / peptidyl-tyrosine phosphorylation / peptidyl-serine phosphorylation / protein tyrosine kinase activity / learning or memory / non-specific serine/threonine protein kinase / protein phosphorylation / negative regulation of gene expression / protein serine kinase activity / protein serine/threonine kinase activity / neuronal cell body / positive regulation of gene expression / perinuclear region of cytoplasm / signal transduction / nucleoplasm / ATP binding / nucleus / cytosol 類似検索 - 分子機能
Tau-tubulin kinase 1, catalytic domain / : / Protein kinase domain / Serine/Threonine protein kinases, catalytic domain / Protein kinase, ATP binding site / Protein kinases ATP-binding region signature. / Protein kinase domain profile. / Protein kinase domain / Protein kinase-like domain superfamily 類似検索 - ドメイン・相同性
解像度: 2.8→48.686 Å / Cor.coef. Fo:Fc: 0.947 / Cor.coef. Fo:Fc free: 0.932 / SU B: 14.942 / SU ML: 0.216 / 交差検証法: FREE R-VALUE / ESU R: 0.329 / ESU R Free: 0.246 詳細: Hydrogens have been used if present in the input file
Rfactor
反射数
%反射
Rfree
0.2285
1887
5.185 %
Rwork
0.2
34506
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all
0.201
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obs
-
36393
99.47 %
溶媒の処理
イオンプローブ半径: 0.8 Å / 減衰半径: 0.8 Å / VDWプローブ半径: 1.2 Å / 溶媒モデル: MASK BULK SOLVENT