解像度: 1.6→63.2 Å / Cor.coef. Fo:Fc: 0.972 / Cor.coef. Fo:Fc free: 0.954 / SU B: 5.835 / SU ML: 0.084 / 交差検証法: THROUGHOUT / σ(F): 0 / ESU R: 0.088 / ESU R Free: 0.085 詳細: HYDROGENS HAVE BEEN ADDED IN THE RIDING POSITIONS U VALUES : REFINED INDIVIDUALLY THE (DIMETHYLAMINO)NAPHTHALENE GROUPS OF THE LIGAND HAVE NOT BEEN MODELLED AS THERE IS INSUFFICIENT DENSITY, ...詳細: HYDROGENS HAVE BEEN ADDED IN THE RIDING POSITIONS U VALUES : REFINED INDIVIDUALLY THE (DIMETHYLAMINO)NAPHTHALENE GROUPS OF THE LIGAND HAVE NOT BEEN MODELLED AS THERE IS INSUFFICIENT DENSITY, AND THE SULFONYL GROUP IS ONLY MODELLED IN THE ACTIVE SITES OF MOLECULES A AND D. THE HYDROCARBON TAILS OF THE LIGAND MOLECULES ARE EITHER MODELLED WITH LOWERED OCCUPANCY ATOMS OR WITHOUT SOME ATOMS. IN SOME OF THE MOLECULES THE LOOPS BETWEEN THR432 AND GLU449 HAVE BEEN MODELLED AT REDUCED OCCUPANCY OR WITH CHAIN BREAKS WHERE RESIDUES COULD NOT BE PLACED.