登録情報 データベース : PDB / ID : 4lys 構造の表示 ダウンロードとリンクタイトル Crystal Structure of BRD4(1) bound to Colchiceine 要素Bromodomain-containing protein 4 詳細 キーワード PROTEIN BINDING/INHIBITOR / bromodomain / BRD4 inhibitor / epigenetic reader protein / acetylated lysine / histone tail / nucleus / PROTEIN BINDING-INHIBITOR complex機能・相同性 機能・相同性情報分子機能 ドメイン・相同性 構成要素
RNA polymerase II C-terminal domain binding / negative regulation of DNA damage checkpoint / P-TEFb complex binding / negative regulation by host of viral transcription / positive regulation of T-helper 17 cell lineage commitment / positive regulation of G2/M transition of mitotic cell cycle / histone reader activity / RNA polymerase II CTD heptapeptide repeat kinase activity / condensed nuclear chromosome / positive regulation of transcription elongation by RNA polymerase II ... RNA polymerase II C-terminal domain binding / negative regulation of DNA damage checkpoint / P-TEFb complex binding / negative regulation by host of viral transcription / positive regulation of T-helper 17 cell lineage commitment / positive regulation of G2/M transition of mitotic cell cycle / histone reader activity / RNA polymerase II CTD heptapeptide repeat kinase activity / condensed nuclear chromosome / positive regulation of transcription elongation by RNA polymerase II / transcription coregulator activity / lysine-acetylated histone binding / p53 binding / chromosome / regulation of inflammatory response / positive regulation of canonical NF-kappaB signal transduction / Potential therapeutics for SARS / transcription coactivator activity / transcription cis-regulatory region binding / chromatin remodeling / DNA damage response / chromatin binding / regulation of transcription by RNA polymerase II / positive regulation of DNA-templated transcription / enzyme binding / positive regulation of transcription by RNA polymerase II / nucleoplasm / nucleus 類似検索 - 分子機能 Bromodomain protein 4, C-terminal / C-terminal domain of bromodomain protein 4 / NET domain superfamily / NET domain profile. / Brdt, bromodomain, repeat II / : / Brdt, bromodomain, repeat I / NET domain / Bromodomain extra-terminal - transcription regulation / Bromodomain-like ... Bromodomain protein 4, C-terminal / C-terminal domain of bromodomain protein 4 / NET domain superfamily / NET domain profile. / Brdt, bromodomain, repeat II / : / Brdt, bromodomain, repeat I / NET domain / Bromodomain extra-terminal - transcription regulation / Bromodomain-like / Histone Acetyltransferase; Chain A / Bromodomain, conserved site / Bromodomain signature. / Bromodomain / Bromodomain profile. / bromo domain / Bromodomain / Bromodomain-like superfamily / Up-down Bundle / Mainly Alpha 類似検索 - ドメイン・相同性生物種 Homo sapiens (ヒト)手法 X線回折 / 分子置換 / 解像度 : 1.83 Å 詳細データ登録者 Wohlwend, D. / Gerhardt, S. / Einsle, O. 引用ジャーナル : Angew.Chem.Int.Ed.Engl. / 年 : 2013タイトル : 4-Acyl pyrroles: mimicking acetylated lysines in histone code reading.著者 : Lucas, X. / Wohlwend, D. / Hugle, M. / Schmidtkunz, K. / Gerhardt, S. / Schule, R. / Jung, M. / Einsle, O. / Gunther, S. 履歴 登録 2013年7月31日 登録サイト : RCSB / 処理サイト : RCSB改定 1.0 2014年1月15日 Provider : repository / タイプ : Initial release改定 1.1 2014年1月29日 Group : Non-polymer description / Structure summary
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