登録情報 データベース : PDB / ID : 7z3k 構造の表示 ダウンロードとリンクタイトル Autotaxin in complex with orthosteric site-binder CpdA 要素Isoform 2 of Ectonucleotide pyrophosphatase/phosphodiesterase family member 2 詳細 キーワード HYDROLASE / ENPP2 / lysophosphatidic acid / lipid chaperone / / pulmonary fibrosis / GPCR / drug development / small-molecule inhibitor機能・相同性 機能・相同性情報分子機能 ドメイン・相同性 構成要素
response to polycyclic arene / alkylglycerophosphoethanolamine phosphodiesterase / sphingolipid catabolic process / phospholipase D / phospholipid catabolic process / phosphatidylcholine catabolic process / phospholipase D activity / positive regulation of lamellipodium morphogenesis / lysophospholipase activity / phosphodiesterase I activity ... response to polycyclic arene / alkylglycerophosphoethanolamine phosphodiesterase / sphingolipid catabolic process / phospholipase D / phospholipid catabolic process / phosphatidylcholine catabolic process / phospholipase D activity / positive regulation of lamellipodium morphogenesis / lysophospholipase activity / phosphodiesterase I activity / scavenger receptor activity / alkylglycerophosphoethanolamine phosphodiesterase activity / polysaccharide binding / negative regulation of cell-matrix adhesion / positive regulation of oligodendrocyte differentiation / positive regulation of epithelial cell migration / positive regulation of focal adhesion assembly / estrous cycle / phospholipid metabolic process / positive regulation of substrate adhesion-dependent cell spreading / cellular response to cadmium ion / regulation of cell migration / cell chemotaxis / cellular response to estradiol stimulus / positive regulation of peptidyl-tyrosine phosphorylation / nucleic acid binding / immune response / calcium ion binding / positive regulation of cell population proliferation / extracellular space / zinc ion binding 類似検索 - 分子機能 Somatomedin B domain, chordata / Somatomedin B -like domains / Somatomedin B domain / Somatomedin B-like domain superfamily / Somatomedin B domain / Somatomedin B domain (SMB) signature. / Somatomedin B (SMB) domain profile. / Type I phosphodiesterase/nucleotide pyrophosphatase/phosphate transferase / Type I phosphodiesterase / nucleotide pyrophosphatase / Extracellular Endonuclease, subunit A ... Somatomedin B domain, chordata / Somatomedin B -like domains / Somatomedin B domain / Somatomedin B-like domain superfamily / Somatomedin B domain / Somatomedin B domain (SMB) signature. / Somatomedin B (SMB) domain profile. / Type I phosphodiesterase/nucleotide pyrophosphatase/phosphate transferase / Type I phosphodiesterase / nucleotide pyrophosphatase / Extracellular Endonuclease, subunit A / DNA/RNA non-specific endonuclease / DNA/RNA non-specific endonuclease / DNA/RNA non-specific endonuclease / DNA/RNA non-specific endonuclease / DNA/RNA non-specific endonuclease superfamily / His-Me finger superfamily / Alkaline-phosphatase-like, core domain superfamily 類似検索 - ドメイン・相同性 7alpha-hydroxycholesterol / Chem-IA0 / IODIDE ION / THIOCYANATE ION / Autotaxin 類似検索 - 構成要素生物種 Rattus norvegicus (ドブネズミ)手法 X線回折 / シンクロトロン / 分子置換 / 解像度 : 2 Å 詳細データ登録者 Salgado-Polo, F. / Ford, P. / Heckmann, B. / Perrakis, A. 資金援助 1件 詳細 詳細を隠す 引用ジャーナル : Cell Chem Biol / 年 : 2023タイトル : Autotaxin facilitates selective LPA receptor signaling.著者 : Salgado-Polo, F. / Borza, R. / Matsoukas, M.T. / Marsais, F. / Jagerschmidt, C. / Waeckel, L. / Moolenaar, W.H. / Ford, P. / Heckmann, B. / Perrakis, A. 履歴 登録 2022年3月2日 登録サイト : PDBE / 処理サイト : PDBE改定 1.0 2023年1月25日 Provider : repository / タイプ : Initial release改定 1.1 2023年2月1日 Group : Database references / カテゴリ : citationItem : _citation.journal_volume / _citation.page_first / _citation.page_last改定 1.2 2024年2月7日 Group : Data collection / Refinement descriptionカテゴリ : chem_comp_atom / chem_comp_bond / pdbx_initial_refinement_model
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