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Title | A Structural Comparison of Oral SARS-CoV-2 Drug Candidate Ibuzatrelvir Complexed with the Main Protease (Mpro) of SARS-CoV-2 and MERS-CoV |
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Journal, issue, pages | Jacs Au, Year 2024 |
Publish date | May 5, 2024 (structure data deposition date) |
Authors | Chen, P. / Van Oers, T.J. / Arutyunova, E. / Fischer, C. / Wang, C. / Lamer, T. / van Belkum, M.J. / Young, H.S. / Vederas, J.C. / Lemieux, M.J. |
External links | Jacs Au / Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.5 - 2 Å |
Structure data | PDB-9boo: PDB-9bpf: |
Chemicals |
ChemComp-YDL: ChemComp-HOH: |
Source |
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Keywords | VIRAL PROTEIN / PF-07817883 / nsp5 / Main protease / MERS-CoV / SARS-CoV-2 / inhibitor / inhibitory activity |