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-Structure paper
Title | Discovery and Hit to Lead Optimization of Macrocyclic Peptides as Novel Tropomyosin Receptor Kinase A Antagonists |
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Journal, issue, pages | J. Med. Chem., Year 2024 |
Publish date | Mar 25, 2024 (structure data deposition date) |
![]() | Yamada, T. / Mihara, K. / Ueda, T. / Yamauchi, D. / Shimizu, M. / Ando, A. / Mayumi, K. / Nakata, Z. / Mikamiyama, H. |
![]() | ![]() |
Methods | X-ray diffraction |
Resolution | 2.26 - 2.34 Å |
Structure data | ![]() PDB-8ytd: ![]() PDB-8yte: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-GM1: |
Source |
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![]() | TRANSFERASE / cyclic peptide |