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-Structure paper
Title | Discovery of Novel NLRP3 Inflammasome Inhibitors Composed of an Oxazole Scaffold Bearing an Acylsulfamide. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 14, Page 1833-1838, Year 2023 |
Publish date | Oct 17, 2023 (structure data deposition date) |
![]() | Ohba, Y. / Adachi, K. / Furukawa, T. / Nishimaru, T. / Sakurai, K. / Masuo, R. / Inami, T. / Orita, T. / Akai, S. / Adachi, T. ...Ohba, Y. / Adachi, K. / Furukawa, T. / Nishimaru, T. / Sakurai, K. / Masuo, R. / Inami, T. / Orita, T. / Akai, S. / Adachi, T. / Usui, K. / Hamada, Y. / Mori, M. / Kurimoto, T. / Wakashima, T. / Akiyama, Y. / Miyazaki, S. / Noji, S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.7 Å |
Structure data | ![]() PDB-8wsm: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ADP: ![]() ChemComp-XE3: ![]() ChemComp-HOH: |
Source |
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![]() | IMMUNE SYSTEM / inflammasome |