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-Structure paper
Title | Discovery of a brain-permeable bromodomain and extra terminal domain (BET) inhibitor with selectivity for BD1 for the treatment of multiple sclerosis. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 265, Page 116080-116080, Year 2023 |
Publish date | Sep 25, 2023 (structure data deposition date) |
![]() | Chen, X. / Wu, T. / Du, Z. / Kang, W. / Xu, R. / Meng, F. / Liu, C. / Chen, Y. / Bao, Q. / Shen, J. ...Chen, X. / Wu, T. / Du, Z. / Kang, W. / Xu, R. / Meng, F. / Liu, C. / Chen, Y. / Bao, Q. / Shen, J. / You, Q. / Cao, D. / Jiang, Z. / Guo, X. |
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Methods | X-ray diffraction |
Resolution | 1.4 Å |
Structure data | ![]() PDB-8wiu: |
Chemicals | ![]() ChemComp-WPR: ![]() ChemComp-HOH: |
Source |
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![]() | DNA BINDING PROTEIN / binds acetylated lysine residues |