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-Structure paper
Title | Accurate Characterization of Binding Kinetics and Allosteric Mechanisms for the HSP90 Chaperone Inhibitors Using AI-Augmented Integrative Biophysical Studies. |
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Journal, issue, pages | Jacs Au, Vol. 4, Page 1632-1645, Year 2024 |
Publish date | Aug 22, 2023 (structure data deposition date) |
![]() | Xu, C. / Zhang, X. / Zhao, L. / Verkhivker, G.M. / Bai, F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.55 - 2.25 Å |
Structure data | ![]() PDB-8ki4: ![]() PDB-8w4v: ![]() PDB-8w8k: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]() ChemComp-MG: ![]()
ChemComp-Q9O: ![]() ChemComp-TUH: |
Source |
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![]() | CHAPERONE / HSP90 / ATPase / NTD / Complex / Inhibitor |