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-Structure paper
Title | Combining VPS34 inhibitors with STING agonists enhances type I interferon signaling and anti-tumor efficacy. |
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Journal, issue, pages | Mol Oncol, Year 2024 |
Publish date | Feb 7, 2024 (structure data deposition date) |
![]() | Yu, Y. / Bogdan, M. / Noman, M.Z. / Parpal, S. / Bartolini, E. / Van Moer, K. / Kleinendorst, S.C. / Bilgrav Saether, K. / Tresaugues, L. / Silvander, C. ...Yu, Y. / Bogdan, M. / Noman, M.Z. / Parpal, S. / Bartolini, E. / Van Moer, K. / Kleinendorst, S.C. / Bilgrav Saether, K. / Tresaugues, L. / Silvander, C. / Lindstrom, J. / Simeon, J. / Timson, M.J. / Al-Hashimi, H. / Smith, B.D. / Flynn, D.L. / Alexeyenko, A. / Viklund, J. / Andersson, M. / Martinsson, J. / Pokrovskaja Tamm, K. / De Milito, A. / Janji, B. |
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Methods | X-ray diffraction |
Resolution | 2.06 Å |
Structure data | ![]() PDB-8rxr: |
Chemicals | ![]() PDB-1h4e: ![]() ChemComp-PEG: ![]() ChemComp-IMD: ![]() ChemComp-DMS: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN / Inhibitor / Complex / Kinase / Autophagy / Drug Discovery / Signaling |