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-Structure paper
Title | Discovery and chemical optimisation of a Potent, Bi-cyclic (Bicycle) Antimicrobial Inhibitor of Escherichia coli PBP3 |
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Journal, issue, pages | To Be Published |
Publish date | Jan 29, 2024 (structure data deposition date) |
![]() | Rowland, C.E. / Newman, H. / Martin, T.T. / Dods, R. / Bournakas, N. / Wagstaff, J.M. / Lewis, N. / Stanway, S.J. / Blamforth, M. / Kessler, C. ...Rowland, C.E. / Newman, H. / Martin, T.T. / Dods, R. / Bournakas, N. / Wagstaff, J.M. / Lewis, N. / Stanway, S.J. / Blamforth, M. / Kessler, C. / van Rietschoten, K. / Bellini, D. / Roper, D.I. / Lloyd, A.J. / Dowson, C.G. / Skynner, M.J. / Beswick, P. / Dawson, M. |
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Methods | X-ray diffraction |
Resolution | 1.52 Å |
Structure data | ![]() PDB-8rtz: |
Chemicals | ![]() ChemComp-29N: ![]() ChemComp-HOH: |
Source |
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