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-Structure paper
Title | Bridging the maytansine and vinca sites: Cryptophycins target beta-tubulin's T5-loop. |
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Journal, issue, pages | J. Biol. Chem., Vol. 300, Page 107363-107363, Year 2024 |
Publish date | Nov 21, 2023 (structure data deposition date) |
![]() | Abel, A.C. / Muhlethaler, T. / Dessin, C. / Schachtsiek, T. / Sammet, B. / Sharpe, T. / Steinmetz, M.O. / Sewald, N. / Prota, A.E. |
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Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-8r67: |
Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-CA: ![]() ChemComp-GDP: ![]() ChemComp-IMD: ![]() ChemComp-MES: ![]() ChemComp-GOL: ![]()
ChemComp-Y74: ![]() ChemComp-ACP: ![]() ChemComp-HOH: |
Source |
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![]() | CELL CYCLE / TUBULIN FOLD / CYTOSKELETON / MICROTUBULE |