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-Structure paper
Title | What doesn't fit is made to fit: Pim-1 kinase adapts to the configuration of stilbene-based inhibitors. |
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Journal, issue, pages | Arch Pharm, Vol. 357, Page e2400094-e2400094, Year 2024 |
Publish date | Nov 1, 2023 (structure data deposition date) |
![]() | Hochban, P.M.M. / Heyder, L. / Heine, A. / Diederich, W.E. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.89 - 2.45 Å |
Structure data | ![]() PDB-8r10: ![]() PDB-8r18: ![]() PDB-8r1n: ![]() PDB-8r1p: ![]() PDB-8r1t: |
Chemicals | ![]()
ChemComp-XGQ: ![]() ChemComp-HOH: ![]() ChemComp-GOL: ![]()
ChemComp-XGK: ![]() ChemComp-EDO: ![]()
ChemComp-XIT: ![]()
ChemComp-XIP: ![]()
ChemComp-XIJ: |
Source |
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![]() | TRANSFERASE / SERINE KINASE / KINASE / COMPLEX / PIM1 / PIM / PIM-1 / INHIBITOR / TUMORIGENISIS / CANCER / PIMTIDE / PROTO ONCOGEN / ATP / PHOSPHORYLATION / APOPTOSIS / CELL CYCLE |