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-Structure paper
Title | Targeting a key protein-protein interaction surface on mitogen-activated protein kinases by a Michael acceptor-based cyclic warhead scaffold |
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Journal, issue, pages | To Be Published |
Publish date | Jul 13, 2023 (structure data deposition date) |
![]() | Sok, P. / Poti, A. / Balint, D. / Soos, T. / Remenyi, A. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.65 - 2.55 Å |
Structure data | ![]() PDB-8psr: ![]() PDB-8pst: ![]() PDB-8psw: ![]() PDB-8psy: ![]() PDB-8pt0: ![]() PDB-8pt1: ![]() PDB-8pt3: ![]() PDB-8pt5: |
Chemicals | ![]() ChemComp-ANP: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-AN2: ![]()
ChemComp-DC6: ![]()
ChemComp-D2I: ![]()
ChemComp-EI0: ![]()
ChemComp-EAI: ![]()
ChemComp-E2A: ![]()
ChemComp-D7O: ![]()
ChemComp-D5R: |
Source |
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![]() | SIGNALING PROTEIN / MAPK kinase / MAPK / inhibitor / covalent / ERK2 / Michael acceptor warhead |