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-Structure paper
Title | Structural insight into the macrocyclic inhibitor TPX-0022 of c-Met and c-Src. |
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Journal, issue, pages | Comput Struct Biotechnol J, Vol. 21, Page 5712-5718, Year 2023 |
Publish date | Jul 26, 2023 (structure data deposition date) |
![]() | Qu, L. / Lin, H. / Dai, S. / Guo, M. / Chen, X. / Jiang, L. / Zhang, H. / Li, M. / Liang, X. / Chen, Z. ...Qu, L. / Lin, H. / Dai, S. / Guo, M. / Chen, X. / Jiang, L. / Zhang, H. / Li, M. / Liang, X. / Chen, Z. / Wei, H. / Chen, Y. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.67 - 2.8 Å |
Structure data | ![]() PDB-8k78: ![]() PDB-8k79: |
Chemicals | ![]()
ChemComp-IYC: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / cMET / TPX-0022 / SRC |