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-Structure paper
Title | Structure-based design and synthesis of BML284 derivatives: A novel class of colchicine-site noncovalent tubulin degradation agents. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 268, Page 116265-116265, Year 2024 |
Publish date | May 30, 2023 (structure data deposition date) |
![]() | Zhang, C. / Yan, W. / Liu, Y. / Tang, M. / Teng, Y. / Wang, F. / Hu, X. / Zhao, M. / Yang, J. / Li, Y. |
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Methods | X-ray diffraction |
Resolution | 2.68 - 2.76 Å |
Structure data | ![]() PDB-8jjb: ![]() PDB-8jjc: |
Chemicals | ![]() ChemComp-GTP: ![]() ChemComp-MG: ![]() ChemComp-CA: ![]() ChemComp-MES: ![]()
ChemComp-USI: ![]() ChemComp-GDP: ![]() ChemComp-CL: ![]() ChemComp-ACP: ![]() ChemComp-HOH: ![]()
ChemComp-UPO: |
Source |
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![]() | CELL CYCLE / Microtubule |